反应条件
1: [3H]-Indoleacetic acid With sodium hydride in N,N-dimethyl-formamide T=0°C; 0.5 h; 2: 4-bromomethyl-fluorobenzene in N,N-dimethyl-formamide T=0°C; 1 h; 3: With hydrogenchloride in water; N,N-dimethyl-formamide
参考文献
Xu, Qinyuan; Huang, Li; Liu, Juan; Ma, Liang; Chen, Tao; Chen, Jinying; Peng, Fei; Cao, Dong; Yang, Zhuang; Qiu, Neng; Qiu, Jingxiang; Wang, Guangcheng; Liang, Xiaolin; Peng, Aihua; Xiang, Mingli; Wei, Yuquan; Chen, Lijuan
European Journal of Medicinal Chemistry, 2012 , vol. 52, p. 70 - 81