反应条件
<b>Multi-step reaction with 2 steps<br /> </b>1: 73 percent / K<sub>2</sub>CO<sub>3</sub> / tetrahydrothiophene 1,1-dioxide / 15 h / 140 °C<br />2: 70 percent / (Ph<sub>3</sub>P)4Pd; aq. Na<sub>2</sub>CO<sub>3</sub> / ethanol; toluene / 2 h / Heating<br /> <br />
参考文献
Murugesan; Gu; Stein; Spergel; Mathur; Leith; Liu; Zhang; Bird; Waldron; Marino; Morrison; Webb; Moreland; Barrish Journal of Medicinal Chemistry, 2000 , vol. 43, # 16 p. 3111 - 3117