反应条件
1: 95 percent / NaOH / methanol / 6 h / Heating 2: 1.) Et3N, diphenyl phosphorazidate, 2.) conc. HCl, phenol / 1) reflux, 22.5 h; 2) 110 deg C, 45 h 3: 100 percent / thionyl chloride / 100 h / Heating View Scheme
参考文献
Nesloney, Carey L.; Kelly, Jeffery W.
Journal of Organic Chemistry, 1996 , vol. 61, # 9 p. 3127 - 3137