反应条件
1: Et3N, DPPA / benzene / 1 h / 50 °C 2: 1,2-dichloro-benzene / 1 h / Heating 3: 88 percent / POCl3 / 1 h / Heating 4: 93 percent / 28percent NH4OH / methanol / 48 h / 150 °C 5: 80 percent / sodium bis(2-methoxyethoxy)aluminium hydride / toluene / 0.5 h / Heating View Scheme
参考文献
Yoshioka, Haruyuki; Matsuya, Yuhji; Choshi, Tominari; Sugino, Eiichi; Hibino, Satoshi
Chemical and Pharmaceutical Bulletin, 1996 , vol. 44, # 4 p. 709 - 714