反应条件
1: 95 percent / HCl(g) 2: 1.) Wang resin, Huenig's base, 2.) 3percent Pd(PPh3)4, 2M Na2CO3, 3.) Br2, pyridine / 1.) DMF, 40-50 deg C, 2.) DME, reflux, 3.) DMF, 80-90 deg C, 24 h View Scheme
参考文献
Han, Yongxin; Walker, Shawn D.; Young, Robert N.
Tetrahedron Letters, 1996 , vol. 37, # 16 p. 2703 - 2706