反应条件
1: 31 percent / NaNO3, TFA, Ac2O / 15 h / Ambient temperature
2: 99 percent / DDQ / benzene / 8 h / Heating
View Scheme
参考文献
Chou, M. W.; Heflich, R. H.; Casciano, D. A.; Miller, D. W.; Freeman, J. P.; et al.
Journal of Medicinal Chemistry, 1984 , vol. 27, # 9 p. 1156 - 1161