反应条件
1: NaH / CH2Cl2 / 2.25 h / 0 - 20 °C 2: 1.) PPh3, DEAD / 1.) THF, 10 min, 2.) THF, RT, overnight 3: Bu4NF / tetrahydrofuran View Scheme
参考文献
Zacharie, Boulos; Gagnon, Lyne; Attardo, Giorgio; Connolly, Timothy P.; St-Denis, Yves; Penney, Christopher L.
Journal of Medicinal Chemistry, 1997 , vol. 40, # 18 p. 2883 - 2894