反应条件
1: 76 percent / tetrahydrofuran; diethyl ether / 0.5 h / Ambient temperature 2: 1.) NaH / 1.) THF, 30 min, 2.) THF, 3 h View Scheme
参考文献
Zhang, Lin; Nadzan, Alex M.; Heyman, Richard A.; Love, Deborah L.; Mais, Dale E.; Croston, Glenn; Lamph, William W.; Boehm, Marcus F.
Journal of Medicinal Chemistry, 1996 , vol. 39, # 14 p. 2659 - 2663