反应条件
1.1: NaH / N,N-dimethyl-acetamide / 0.5 h / 20 °C
1.2: 86 percent / N,N-dimethyl-acetamide / 6 h / 20 °C
2.1: 92 percent / KOH / 2-methyl-propan-2-ol / 4 h / 80 °C
View Scheme
参考文献
Mano, Takashi; Stevens, Rodney W.; Nakao, Kazunari; Okumura, Yoshiyuki; Kawamura, Kiyoshi; Ando, Akemi; Matsuoka, Yoko
Synthesis, 2004 , # 16 p. 2625 - 2628