4-碘-1H-吡唑-3-羧酸乙酯合成路线 （共 2 条）
反应条件
ammonium cerium (IV) nitrate; iodine in acetonitrile
T=20°C; 20 h;
参考文献
MERCK SHARP and DOHME CORP.; ADDEX PHARMA S.A.; LIVERTON, Nigel, J.; BOLEA, Christelle; CELANIRE, Sylvain; YUNFU, Luo
Patent: WO2012/8999 A2, 2012 ;
Location in patent: Page/Page column 47; 48 ;
WO 2012/008999 A2
反应条件
1: tetrahydrofuran / 3 h / 20 - 30 °C
2: iodine; ammonium cerium (IV) nitrate / acetonitrile / 20 h / 20 °C
View Scheme
参考文献
MERCK SHARP and DOHME CORP.; ADDEX PHARMA SA; LIVERTON, Nigel, J.; BOLEA, Christelle; CELANIRE, Sylvain; LUO, Yunfu
Patent: WO2012/6760 A1, 2012 ;
WO 2012/006760 A1
