反应条件
1: 20 percent / I2, catechol, 4A molecular sieves / 48 h / Heating 2: 1.) n-BuLi / 1.) THF, -75 deg C, 15 min, 2.) THF, 0 deg C View Scheme
参考文献
Pooley, Charlotte L. F.; Edwards, James P.; Goldman, Mark E.; Wang, Ming-Wei; Marschke, Keith B.; Crombie, Diane L.; Jones, Todd K.
Journal of Medicinal Chemistry, 1998 , vol. 41, # 18 p. 3461 - 3466