5-氟-2-甲氧基苯硼酸合成路线 (共 11 条)
反应条件
sodium carbonate; tetrakis(triphenylphosphine) palladium(0) in ethanol; water; toluene
Heating / reflux;
参考文献
ASTRAZENECA AB; ASTRAZENECA UK LIMITED
Patent: WO2006/21759 A1, 2006 ;
Location in patent: Page/Page column 66 ;
WO 2006/021759 A1