反应条件
1: (S)-1-(6-amino-9H-purin-9-yl) propan-2-ol With Mg(O-t-Bu)2 in N,N-dimethyl-formamide T=20°C; 1 h; Inert atmosphere; 2: diethyl p-toluenesulfonyloxymethylphosphonate in N,N-dimethyl-formamide T=35°C; 20 h; Inert atmosphere;
参考文献
European Journal of Medicinal Chemistry, , vol. 63, p. 869 - 881