2-氨基-1,3-苯并噻唑-6-磺酰胺合成路线 (共 13 条)
反应条件
1: With ammonium thiocyanate in acetic acid T=20°C; 0.5 h; 2: With bromine in acetic acid T=20°C; 64 h; 3: With sodium hydrogencarbonate in water
参考文献
WO2004/11460 A2, ;
Page 59-60 ;
WO 2004/011460 A2
反应条件
bromine in chloroform 0.25 h; Reflux;
参考文献
Sharma, Pawan K.; Chandna, Nisha; Kumar, Surender; Kmar, Pawan; Kumar, Satish; Kaushik, Pawan; Kaushik, Dhirender
Medicinal Chemistry Research, 2012 , vol. 21, # 11 p. 3757 - 3766
反应条件
1: bromine; methanol 2: acetic acid View Scheme
参考文献
Archiv der Pharmazie (Weinheim, Germany), , vol. 279, p. 194,204
反应条件
ammonium hydroxide in acetone 0.0833333 h; Heating;
参考文献
Archiv der Pharmazie und Berichte der Deutschen Pharmazeutischen Gesellschaft, , vol. 302, # 7 p. 511 - 517
反应条件
bromine in acetic acid
参考文献
Pharmazie, , vol. 22, p. 620 - 624
反应条件
bromine; acetic acid
参考文献
J. Chin. chem. Soc., , vol. 15, p. 208,212
Archiv der Pharmazie (Weinheim, Germany), , vol. 279, p. 194,204
Yakugaku Zasshi, , vol. 71, p. 553,554
Chem.Abstr., , p. 4546
参考文献
Archiv der Pharmazie (Weinheim, Germany), , vol. 279, p. 181,186
参考文献
Archiv der Pharmazie (Weinheim, Germany), , vol. 279, p. 194,204
参考文献
J. Chin. chem. Soc., , vol. 15, p. 208,212
反应条件
bromine; acetic acid
参考文献
Letters in Drug Design and Discovery, , vol. 8, # 9 p. 774 - 777