1: 4-aminobutylguanidine sulfate With potassium carbonate in water T=0 - 5°C; 0.166667 h; 2: acryloyl chloride in water; acetone T=5°C; 1 h; 3: With sulfuric acid; potassium carbonate Product distribution / selectivity; more than 3 stages;
参考文献
AMERSHAM BIOSCIENCES AB
Patent: WO2005/40092 A1, 2005 ;
Location in patent: Page/Page column 8 ;