反应条件
1: 83 percent / pyridine / 24 h / Ambient temperature 2: 1.) N,N'-thiocarbonyldiimidazole, 2.) α,α'-azobis(isobutyronitrile), tributyltin hydride / 1.) toluene, MeCN, 80 deg C, 30 min, 2.) MeCN, 80 deg C, 3 h View Scheme
参考文献
Camarasa; Perez-Perez; San-Felix; Balzarini; De Clercq
Journal of Medicinal Chemistry, 1992 , vol. 35, # 15 p. 2721 - 2727