反应条件
1: 1.) Et4NOAc, 2.) K2CO3, 3.) NEt3
2: 83 percent / N-methylmorpholine N-oxide, tetrapropylammonium per-ruthenate / CH2Cl2
View Scheme
参考文献
ASTRAZENECA AB; ASTRAZENECA UK LIMITED; MCGUIRE, Helen; BIST, Shanta; BIFULCO, Neil; ZHAO, Liang; WU, Ye; HUYNH, Hoan; XIONG, Hui; COMITA-PREVOIR, Janelle; DUSSAULT, Daemian; GENG, Bolin; CHEN, Brendan; DURAND-REVILLE, Thomas; GULER, Satenig
Patent: WO2013/150296 A1, 2013 ;