反应条件
1: benzylamine, diethylamine
2: SOCl2 / 2 h / Ambient temperature
3: H2, sodium formate / 5percent Pd/C / tetrahydrofuran; methanol / 6 h / Ambient temperature
View Scheme
参考文献
Trani; Dallanoce; Ferrari; Goldstein; Ripamonti; Ciabatti
Farmaco, 1996 , vol. 51, # 7 p. 503 - 512