1: in DMF (N,N-dimethyl-formamide)
T=20°C; 16 h;
2: With sodium hydride in dimethyl sulfoxide
T=20°C; 1 h;
参考文献
Monia, Brett P.; Freier, Susan M.; Manoharan, Muthiah; Gaarde, William A.; Griffey, Richard H.; Swayze, Eric E.; Bennett, C. Frank
Patent: US2005/130924 A1, 2005 ;
Location in patent: Page/Page column 19; 20 ;