1: m-C6H4BrBCl2 With i -Pr2Zn in diethyl ether T=25°C; 2 h; 2: in tetrahydrofuran T=-30°C; 0.166667 h; 3: allyl bromide in tetrahydrofuran T=20°C; Further stages.;
参考文献
Hupe, Eike; Calaza, M. Isabel; Knochel, Paul
Chemical Communications, 2002 , # 13 p. 1390 - 1391
1: With 9-borabicyclo[3.3.1]nonane dimer in tetrahydrofuran
T=20°C;
2: With sodium hydroxide; dihydrogen peroxide in tetrahydrofuran; water
T=20°C; 4 h; Cooling with ice;
参考文献
ALLERGAN, INC.
Patent: WO2009/6370 A1, 2009 ;
Location in patent: Page/Page column 49 ;
WO 2009/006370 A1