反应条件
1: 64 percent / H2 / PtO2 / methanol / 0.5 h / 1551.4 Torr 2: 11 percent / Et3N, HgCl2 / dimethylformamide / 1.) 5 deg C, 0.5 h, 2.) RT, 18 h View Scheme
参考文献
Chand, Pooran; Babu, Yarlagadda S.; Bantia, Shanta; Chu, Naiming; Cole, L. Brent; Kotian, Pravin L.; Laver, W. Graeme; Montgomery, John A.; Pathak, Ved P.; Petty, Sandra L.; Shrout, David P.; Walsh, David A.; Walsh, Gerald M.
Journal of Medicinal Chemistry, 1997 , vol. 40, # 25 p. 4030 - 4052