反应条件
1: CH2Cl2 / 1 h / Heating
2: CH2Cl2 / 1.) 0 deg C, 30 min, 2.) RT, 1 h
3: 2 N aq. NaOH / 2 h
View Scheme
参考文献
Leone-Bay, Andrea; Paton, Duncan R.; Freeman, John; Lercara, Christine; O'Toole, Doris; Gschneidner, David; Wang, Eric; Harris, Elizabeth; Rosado, Connie; Rivera, Theresa; DeVincent, Aldonna; Tai, Monica; Mercogliano, Frank; Agarwal, Rajesh; Leipold, Harry; Baughman, Robert A.
Journal of Medicinal Chemistry, 1998 , vol. 41, # 7 p. 1163 - 1171