3-(2-甲基-1H-咪唑)苯胺合成路线 (共 1 条)
反应条件
8-hydroxy-quinoline; potassium carbonate; copper(l) iodide in dimethyl sulfoxide T=125 - 130°C; Ullmann Coupling;
参考文献
DUPONT PHARMACEUTICALS COMPANY
Patent: WO2002/8199 A2, 2002 ;
Location in patent: Page 32 ;
WO 02/08199 A2