3-{[(4-氯-3-甲基-5-异噁唑)氨基]磺酰基}-2-噻吩羧酸甲酯合成路线 (共 2 条)
反应条件
sodium hydride 1.) THF, 10 min, 2.) THF, RT, 4 h; Multistep reaction;
参考文献
AUSPEX PHARMACEUTICALS, INC.
Patent: US2008/255036 A1, 2008 ;
Location in patent: Page/Page column 65-66 ;
US 20080255036 A1
参考文献
Texas Biotechnology Corp.
Patent: US6342610 B2, 2002 ;
Location in patent: Page column 100 ;
US 6342610 B2