5-(哌嗪-1-基)-1H-吲哚合成路线 (共 4 条)
反应条件
1: With lithium aluminium tetrahydride in tetrahydrofuran 2: With hydrogenchloride; hydrogen; palladium dihydroxide in ethanol; water P=2280.15 Torr; 65 h;
参考文献
EP1396487 A1, ;
Page 15 ;
反应条件
ammonium formate; palladium on activated carbon 0.75 h; Heating / reflux;
参考文献
US2007/43058 A1, ;
Page/Page column 7 ;
US 20070043058 A1
反应条件
sodium carbonate in hydrogenchloride; ethanol
参考文献
Merck Sharpe and Dohme Ltd.
Patent: US5432177 A1, 1995 ;
反应条件
trifluoroacetic acid in dichloromethane T=20°C; 2 h; Inert atmosphere;
参考文献
WAYNE STATE UNIVERSITY; DUTTA, Aloke, K.
Patent: WO2014/85600 A1, 2014 ;
Location in patent: Page/Page column 00073 ;