反应条件
1: 96 percent / Et3N, diphenyl phosphorazidate / toluene / 3 h / Heating 2: 39 percent / FeCl3 / 1,2-dichloro-ethane View Scheme
参考文献
Fevig, Thomas L.; Bowen, S. Marc; Janowick, David A.; Jones, Bryan K.; Munson, H. Randall; Ohlweiler, David F.; Thomas, Craig E.
Journal of Medicinal Chemistry, 1996 , vol. 39, # 25 p. 4988 - 4996