反应条件
1: SOCl2 / toluene / RT, 30 min then 55 deg C, 1 h 2: 70 percent / K2CO3, NaI / acetonitrile / 24 h / Heating 3: 83 percent / KOH / methanol; H2O / Heating View Scheme
参考文献
Ahmad, Youssef El; Laurent, Elisabeth; Maillet, Philippe; Talab, Akram; Teste, Jean Francois; Dokhan, Raymond; Tran, Gilles; Ollivier, Roland
Journal of Medicinal Chemistry, 1997 , vol. 40, # 6 p. 952 - 960