1: trifluoroacetic acid / dichloromethane / 2 h
2: 1-hydroxy-pyrrolidine-2,5-dione; triethylamine; diisopropyl-carbodiimide / dichloromethane / 16 h
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参考文献
Crielaard, Bart J.; Van Der Wal, Steffen; Le, Huong Thu; Bode, Alois T.L.; Lammers, Twan; Hennink, Wim E.; Schiffelers, Raymond M.; Fens, Marcel H.A.M.; Storm, Gert
European Journal of Pharmaceutical Sciences, 2012 , vol. 45, # 4 p. 429 - 435