1: diethyl malonate With sodium hydride in various solvent(s) T=20°C; 1 h; 2: 1-bromo-4-chloro-butane in various solvent(s) T=20°C; 3 h; Further stages.;
参考文献
Asaki, Tetsuo; Aoki, Tomiyoshi; Hamamoto, Taisuke; Sugiyama, Yukiteru; Ohmachi, Shinji; Kuwabara, Kenji; Murakami, Kohji; Todo, Makoto
Bioorganic and Medicinal Chemistry, 2008 , vol. 16, # 2 p. 981 - 994