反应条件
1: 87 percent / 1N HCl / tetrahydrofuran / 4 h / 0 °C
2: LiOH, LiBr, n-Bu4NBr / acetonitrile / 1 h / Ambient temperature
View Scheme
参考文献
Sagan, Sandrine; Josien, Hubert; Karoyan, Philippe; Brunissen, Alie; Chassaing, Gerard; Lavielle, Solange
Bioorganic and Medicinal Chemistry, 1996 , vol. 4, # 12 p. 2167 - 2178