反应条件
sodium hydride
1.) DMF, 50 deg C, 30 min, 2.) DMF, RT, 1.5 h; Yield given. Multistep reaction;
参考文献
Cywin, Charles L.; Klunder, Janice M.; Hoermann, MaryAnn; Brickwood, Janice R.; David, Eva; Grob, Peter M.; Schwartz, Racheline; Pauletti, Daniel; Barringer, Kevin J.; Shih, Cheng-Kon; Sorge, Christopher L.; Erickson, David A.; Joseph, David P.; Hattox, Susan E.
Journal of Medicinal Chemistry, 1998 , vol. 41, # 16 p. 2972 - 2984