1: 70 percent / Et3N; 3-ethyl-5-(2-hydroxyethyl)-4-methylthiazolium bromide / ethanol / 20 h / 75 - 80 °C 2: 90 percent / aq. Oxone(R) / methanol / 2 h / 25 °C 3: 85 percent / p-toluenesulfonic acid / toluene / 20 h / Heating View Scheme
参考文献
Khanna, Ish K.; Weier, Richard M.; Yu, Yi; Collins, Paul W.; Miyashiro, Julie M.; Koboldt, Carol M.; Veenhuizen, Amy W.; Currie, Jerry L.; Seibert, Karen; Isakson, Peter C.
Journal of Medicinal Chemistry, 1997 , vol. 40, # 11 p. 1619 - 1633
1: 90 percent / aq. Oxone(R) / methanol / 2 h / 25 °C 2: 85 percent / p-toluenesulfonic acid / toluene / 20 h / Heating View Scheme
参考文献
Khanna, Ish K.; Weier, Richard M.; Yu, Yi; Collins, Paul W.; Miyashiro, Julie M.; Koboldt, Carol M.; Veenhuizen, Amy W.; Currie, Jerry L.; Seibert, Karen; Isakson, Peter C.
Journal of Medicinal Chemistry, 1997 , vol. 40, # 11 p. 1619 - 1633
