1: With hydrogenchloride in 1,4-dioxane; methanol T=0 - 20°C; 2: With ammonia in methanol
参考文献
CANCER RESEARCH TECHNOLOGY LIMITED; McDONALD, Edward; BLAGG, Julian; PICHOWICZ, Mark; CRUMPLER, Simon Ross
Patent: WO2010/41054 A1, 2010 ;
Location in patent: Page/Page column 32 ;