(3R,4S)-1-(4-氟苯基)-3-[(3S)-3-乙酰氧基-3-(4-氟苯基)丙基]-4-(4-羟基苯基)-2-氮杂环丁酮合成路线 (共 1 条)
反应条件
aluminum oxide in dichloromethane 0.05 h; microwave irradiation;
参考文献
Kvaerno, Lisbet; Ritter, Tobias; Werder, Moritz; Hauser, Helmut; Carreira, Erick M.
Angewandte Chemie - International Edition, 2004 , vol. 43, # 35 p. 4653 - 4656