反应条件
1: 92 percent / aq. HCl / acetone / 1 h / 25 °C
2: 91 percent / CrO3, H2SO4 / acetone / 0.17 h / 0 - 5 °C
3: 80.3 percent / TsOH*H2O, formic acid / 7 h / 50 - 60 °C
View Scheme
参考文献
Gao, Hongwu; Su, Xiangdong; Li, Zhensu
Steroids, 1997 , vol. 62, # 5 p. 398 - 402