4-(N,N-dimethlyamino)pyridine; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride in dichloromethane T=23°C; 3 h;
参考文献
Tatlock, John H.; Linton, M. Angelica; Hou, Xinjun J.; Kissinger, Charles R.; Pelletier, Laura A.; Showalter, Richard E.; Tempczyk, Anna; Villafranca, J. Ernest
Bioorganic and Medicinal Chemistry Letters, 1997 , vol. 7, # 8 p. 1007 - 1012