反应条件
1: (4-bromo-thiophen-2-yl)-methanol With sodium hydride; dimethyl sulfoxide 1 h; 2: 2-amino-N,N,N-trimethyl-9H-purine-6-ylammonium chloride in dimethyl sulfoxide 1 h; Further stages.;
参考文献
Reinhard; Hull; Von der Lieth; Eichhorn; Kliem; Kaina; Wiessler
Journal of Medicinal Chemistry, 2001 , vol. 44, # 24 p. 4050 - 4061