5-溴-1,2,3-噻唑并[1,5-a]吡啶合成路线 （共 7 条）
反应条件
morpholine T=130°C; 3 h;
参考文献
WO2014/8197 A1, ;
Page/Page column 108 ;
反应条件
1: 67 percent / 1 h / 100 °C 2: 94 percent / aq. HCl / 16 h / 80 °C 3: 86 percent / DMSO, (COCl)2, Et3N / CH2Cl2 4: 66 percent 5: 72 percent / Heating View Scheme
参考文献
Tetrahedron, , vol. 53, # 24 p. 8257 - 8268
反应条件
1: 66 percent 2: 72 percent / Heating View Scheme
参考文献
Tetrahedron, , vol. 53, # 24 p. 8257 - 8268
反应条件
1: 86 percent / DMSO, (COCl)2, Et3N / CH2Cl2 2: 66 percent 3: 72 percent / Heating View Scheme
参考文献
Tetrahedron, , vol. 53, # 24 p. 8257 - 8268
反应条件
1: 94 percent / aq. HCl / 16 h / 80 °C 2: 86 percent / DMSO, (COCl)2, Et3N / CH2Cl2 3: 66 percent 4: 72 percent / Heating View Scheme
参考文献
Tetrahedron, , vol. 53, # 24 p. 8257 - 8268
参考文献
Tetrahedron, , vol. 53, # 24 p. 8257 - 8268
参考文献
Tetrahedron, , vol. 53, # 24 p. 8257 - 8268
