1H-吲唑-4-甲酸甲酯合成路线

18583-89-63-氨基-2-甲基苯甲酸甲酯

192945-49-61H-吲唑-4-甲酸甲酯

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US2012/130078 A1, ;

Page/Page column 4-5 ;
US 20120130078 A1

677306-38-61H-吲唑-4-羧酸+

18107-18-1三甲基硅烷化重氮甲烷

192945-49-61H-吲唑-4-甲酸甲酯

参考文献

WO2007/51062 A2, ;

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WO 2007/051062 A2

192945-49-61H-吲唑-4-甲酸甲酯

885271-63-63-溴吲唑-4-羧酸甲酯

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BOEHRINGER INGELHEIM INTERNATIONAL GMBH; BOEHRINGER INGELHEIM PHARMA GMBH and CO. KG
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WO 2009/134666 A1

192945-49-61H-吲唑-4-甲酸甲酯

709608-85-5(1H-吲唑-4-基)甲醇

参考文献

CHEMOCENTRYX, INC.
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WO 2007/051062 A2

192945-49-61H-吲唑-4-甲酸甲酯

677306-38-61H-吲唑-4-羧酸

参考文献

MERCK SHARP and DOHME LIMITED
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WO 2005/028445 A2

192945-49-61H-吲唑-4-甲酸甲酯+

74-88-4甲基碘

1071428-42-61-甲基-1H-吲唑-4-羧酸甲酯

参考文献

Astellas Pharma Inc.
Patent: EP2141147 A1, 2010 ;
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EP 2141147 A1

420-37-1三甲基氧鎓四氟硼酸+

192945-49-61H-吲唑-4-甲酸甲酯

1071428-43-72-甲基-2H-吲唑-4-羧酸甲酯

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Takeda Pharmaceutical Company Limited
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