1: With sodium tetrahydroborate in tetrahydrofuran; water T=0 - 20°C; 61 h; 2: With sodium hydroxide in water 1 h; Heating / reflux; 3: With hydrogenchloride in water
参考文献
VERNALIS (CAMBRIDGE) LIMITED; CANCER RESEARCH TECHNOLOGY LTD; THE INSTITUTE OF CANCER RESEARCH
Patent: WO2004/72051 A1, 2004 ;
Location in patent: Page 38; 39 ;