1: With dimethylsulfide borane complex in tetrahydrofuran 2 h; Heating / reflux; 2: With hydrogenchloride; water in tetrahydrofuran; methanol T=20°C; 0.5 h; 3: With ammonia in methanol
参考文献
PIRAMED LIMITED; THE INSTITUTE OF CANCER RESEARCH
Patent: WO2008/125839 A2, 2008 ;
Location in patent: Page/Page column 44-45 ;
WO 2008/125839 A2