反应条件
1: 1.) methanesulfonyl chloride, triethylamine, 2.) DBU / 1.) CH2Cl2, room temperature, 30 min, 2.) CH2Cl2, room temperature
2: 82 percent / PdCl2(PPh3)2, triethylamine / tetrahydrofuran / 4 h
View Scheme
参考文献
Crousse, Benoit; Alami, Mouad; Linstrumelle, Gerard
Tetrahedron Letters, 1997 , vol. 38, # 30 p. 5297 - 5300