1: With lithium aluminium tetrahydride in tetrahydrofuran 2 h; 2: With water; sodium hydrogencarbonate in tetrahydrofuran T=0°C; Product distribution / selectivity;
参考文献
LEK PHARMACEUTICALS D.D.
Patent: WO2007/147547 A1, 2007 ;
Location in patent: Page/Page column 15 ;
WO 2007/147547 A1