反应条件
1: 2.) HNO3, AcOH
2: HCl / Heating
3: 90 percent / H2 / Pd/C / ethanol
4: 75 percent / SOCl2, DMF
View Scheme
参考文献
Mederski, Werner W.K.R.; Osswald, Mathias; Dorsch, Dieter; Anzali, Soheila; Christadler, Maria; Schmitges, Claus-Jochen; Wilm, Claudia
Bioorganic and Medicinal Chemistry Letters, 1998 , vol. 8, # 1 p. 17 - 22