反应条件
1: 55 percent / Pd(PPh3)4, n-BuNH2, CuI / benzene / 45 °C
2: CsF / methanol
3: Et3N
4: 85 percent / K2CO3 / dimethylformamide / Ambient temperature
5: CDCl3 / 36 h / 30 °C
View Scheme
参考文献
Shain, Jagadish Chandra; Khamrai, Uttam Kumar; Basak, Amit
Tetrahedron Letters, 1997 , vol. 38, # 34 p. 6067 - 6070