反应条件
1: o-toluidine With sodium hydride in N,N-dimethyl-formamide 0.5 h; 2: 2-fluoro-1-nitrobenzene in N,N-dimethyl-formamide 16 h;
参考文献
O'Neill, David J.; Adedoyin, Adedayo; Alfinito, Peter D.; Bray, Jenifer A.; Cosmi, Scott; Deecher, Darlene C.; Fensome, Andrew; Harrison, Jim; Leventhal, Liza; Mann, Charles; McComas, Casey C.; Sullivan, Nicole R.; Spangler, Taylor B.; Uveges, Albert J.; Trybulski, Eugene J.; Whiteside, Garth T.; Zhang, Puwen
Journal of Medicinal Chemistry, 2010 , vol. 53, # 11 p. 4511 - 4521