反应条件
1: N-iodo-succinimide / N,N-dimethyl-formamide / 18 h / 20 °C 2: tetrakis(triphenylphosphine) palladium(0) / 1-methyl-pyrrolidin-2-one / 2 h / 135 °C / |Inert atmosphere 3: water; sulfuric acid / 18 h / 100 °C View Scheme
参考文献
BIOTA EUROPE LTD; TYNDALL, Edward Malcolm; CZAPLEWSKI, Lloyd George; FISHWICK, Colin William Gordon; YULE, Ian Andrew; MITCHELL, Jeffrey Peter; ANDERSON, Kelly Helen; PITT, Gary Robert William
Patent: WO2013/91011 A1, 2013 ;