2’-三氟甲基二苯基-4-羧基 酸合成路线 (共 2 条)
反应条件
potassium permanganate in 1,4-dioxane 2 h; Reflux;
参考文献
AKAAL PHARMA PTY LTD; GILL, Gurmit, S.; GROBELNY, Damian, W.
Patent: WO2010/42998 A1, 2010 ;
Location in patent: Page/Page column 95 ;
WO 2010/042998 A1
反应条件
sodium chlorite; sodium dihydrogenphosphate in water; tert-butyl alcohol T=20°C; 5.5 h;
参考文献
ASTRAZENECA AB
Patent: WO2004/60882 A1, 2004 ;
Location in patent: Page 56-57 ;
WO 2004/060882 A1