甲基4-乙烯基-1H-吡咯-2-羧酸酯合成路线 (共 1 条)
反应条件
potassium carbonate; tris-(dibenzylideneacetone)dipalladium(0); 1,1'-bis-(di-tert-butylphosphino)ferrocene in 1,4-dioxane; water T=95°C; 3 h; Inert atmosphere;
参考文献
Eli Lilly and Company
Patent: US2012/202797 A1, 2012 ;
Location in patent: Page/Page column 5-6 ;
US 20120202797 A1