反应条件
1: 5-methyl-2,4(1H,3H)-pyrimidinedione With N,O-bis-(trimethylsilyl)-acetamide in acetonitrile 12 h; Reflux; 2: propargyl bromide in acetonitrile T=80°C; 16 h; regioselective reaction;
参考文献
Legros, Vanessa; Hamon, Florian; Violeau, Bruno; Turpin, Frederic; Djedaini-Pilard, Florence; Desire, Jerome; Len, Christophe
Synthesis, 2011 , # 2 art. no. P13610SS, p. 235 - 242